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Derniers dépôts
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Nathan Picois, Lizeth Bodero, Pierre T Milbeo, Thierry Brigaud, Grégory Chaume. Bimodal use of chiral α‐Trifluoromethylalanine in Aib Foldamers: study of the position impact towards the helical screw‐sense preference. Chemistry - A European Journal, In press, ⟨10.1002/chem.202400540⟩. ⟨hal-04516499⟩
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Julia Kaffy, Dimitri Brinet, Jean-Louis Soulier, Isabelle Correia, Nicolo Tonali, et al.. Designed Glycopeptidomimetics Disrupt Protein–Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability. Journal of Medicinal Chemistry, 2016, 59 (5), pp.2025-2040. ⟨10.1021/acs.jmedchem.5b01629⟩. ⟨hal-02467871⟩
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Doumet Georges Helou, A. Mauras, Francois Fasquelle, J. S. Lanza, P. M. Loiseau, et al.. Intranasal vaccine from whole Leishmania donovani antigens provides protection and induces specific immune response against visceral leishmaniasis.. PLoS Neglected Tropical Diseases, 2021, PLoS Neglected Tropical Diseases, 15, pp.e0009627. ⟨10.1371/journal.pntd.0009627⟩. ⟨hal-04482585⟩
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Nicolas Duchemin, Adam Skiredj, Justine Mansot, Karine Leblanc, Jean-Jacques Vasseur, et al.. DNA-Templated [2+2] Photocycloaddition: A Straightforward Entry into the Aplysinopsin Family of Natural Products. Angewandte Chemie International Edition, 2018, 57 (36), pp.11786-11791. ⟨10.1002/anie.201806357⟩. ⟨hal-02197152⟩
Mots-clés
Cytotoxicity
Synthetic methods
Constrained amino acids
Antileishmanial
Coupling
Catalysis
Human
Antimitotic
Chemical diversity
Chitosan
Cyclization
Annonaceae
Benthic cyanobacteria
Fluorescence
5-HT 4 receptor
Chemistry
Combretastatin A-4
Chalcones
Leishmania
Biomimetic synthesis
High-resolution mass spectrometry
Aldehydes
Autoanticorps
Biological activity
Antimicrobial activity
Foldamers
Molecular dynamics
Alkyne
Cancer
Conformational analysis
Enynes
Crystallography
Biotransformation
Autoimmune diseases
Alkynylation
Copper
Benzils
Alkaloids
Michael addition
Heterocycles
Capillary electrophoresis
Mass spectrometry
Fluor
Binding site
IsoCA-4
Controlled study
Natural products
Acetogenin
Glycosylation
Environmental neurotoxin
Autoantibodies
Peptidomimetics
Dereplication
Sodium iodide
CXCR4
Hydrostannation
Aggregation
Force-field
DMSO
Conformational ensemble
Apoptosis
Annulations
Biosynthesis
Leishmaniasis
Carbohydrates
Article
Pigments
Binding
Buchwald-Hartwig-Migita coupling
Circular dichroism
Amphidinolide
Annonacin
Palladium
Antiviral
Peptidomimétiques
Hair
Alteration
NMR
Amyloïde
Alkynes
Tubulin
Molecular networking
Antimalarial
Fluorine
Ribavirin
Ilimaquinone
Peptides
Molecular modeling
ACL
Biosynthèse
Alpha-synuclein
Benzofuran
Fluorinated peptides
Archéométrie des matières colorantes
Glycosides
Amyloid
Asymmetric synthesis
Halogenation
Thiosugars
C-nucleoside